科研成果
 

2012年论文

返回
发布日期:2013-01-08


12-18: Copper-catalyzed oxidative trifluoromethylthiolation of aryl boronic acids with TMSCF3 and elemental sulfur

       Chao Chen, Yan Xie, Lingling Chu, Ruo-Wen Wang, Xingang Zhang and Feng-Ling Qing*  

        Angew. Chem. Int. Ed.2012, 51, 2492-2495. DOI: 10.1002/anie.201108663 

  


12-17: Recent advances of trifluoromethylation

       Feng-Ling Qing*

        Chin. J. Org. Chem.2012, 32,815-824. DOI: 10.6023/cjoc1202021


12-16: An improved copper-mediated oxidative trifluoromethylation of terminal alkynes

       Ke Zhang, Xiao-Long Qiu, Yangen Huang, andFeng-Ling Qing*

        Eur. J. Org. Chem.2012,58-61. DOI: 10.1002/ejoc.201101550

12-15: Copper-catalyzed direct C-H oxidative trifluoromethylation of heteroarenes  

       Lingling Chu and Feng-Ling Qing*  

        J. Am. Chem. Soc.2012, 134, 1298-1304. DOI: 10.1021/ja209992w


12-14: Metal-free oxidative trifluoromethylthiolation of terminal alkynes with CF3SiMe3 and elemental sulfur

       Chao Chen, Lingling Chu and Feng-Ling Qing*  

        J. Am.. Chem. Soc.2012, 134, 12454-12457. DOI: 10.1021/ja305801m


12-13: Palladium-catalyzed direct α-arylation of α-fluoroketones: A straightforward route to α-fluoro-α-arylketones

       Chen Guo, Ruo-Wen Wang, Yong Guo, andFeng-Ling Qing*

        J. Fluorine Chem.2012, 133,86-96. DOI: 10.1016/j.jfluchem.2011.08.004


12-12: Coupling of sterically hindered aldehyde with fluorinated synthons: Stereoselective synthesis of fluorinated analogues of salinosporamide A

       Zeng-Hao Chen, Bing-Lin Wang, Andrew J. Kale, Bradley S. Moore, Ruo-Wen Wang, andFeng-Ling Qing*

        J. Fluorine Chem.2012, 136,12-19. DOI: 10.1016/j.jfluchem.2012.01.003


12-11: Palladium catalyzed direct α-arylation of α,α-difluoroketones with aryl bromides

       Chen Guo, Ruo-Wen Wang, andFeng-Ling Qing*

        J. Fluorine Chem.2012, 143,135-142. DOI: 10.1016/j.jfluchem.2012.05.001


12-10: Copper-catalyzed oxidative trifluoromethylation of terminal alkynes and aryl boronic acids using (trifluoromethyl)trimethylsilane

       Xueliang Jiang, Lingling Chu and Feng-Ling Qing*  

        J. Org. Chem.2012, 77, 1251-1257. DOI: 10.1021/jo202566h 


12-9: Sequential electrophilic trifluoromethanesulfanylation-cyclization of tryptamine derivatives: Synthesis of C(3)-trifluoromethanesulfanylated hexahydropyrrolo[2,3-b]indoles

       Yi Yang, Xueliang Jiang and Feng-Ling Qing*  

        J. Org. Chem.2012, 77, 7538-7547. DOI: 10.1021/jo3013385 

12-8: Regio- and diastereoselective nickel-catalyzed allylation of aromatic aldehydes with α-halo-β,β-difluoropropene derivatives

       Xiaowei Lin, Feng Zheng and Feng-Ling Qing*  

        J. Org. Chem.2012, 77, 8696-8704. DOI: 10.1021/jo301688d

  


12-7: Copper-catalyzed oxidative trifluoromethylation of terminal alkenes using nucleophilic CF3SiMe3: Efficient C(sp3)-CF3 bond formationand

       Lingling Chu and Feng-Ling Qing*  

        Org. Lett.2012, 14, 2106-2109. DOI: 10.1021/ol300639a 

  

12-6: Copper-mediated oxidative cross-coupling reaction of terminal alkynes with α-silyldifluoronethylphosphonates: An efficient method for α,α-difluoropropargylphosphonates

       Xueliang Jiang, Lingling Chu and Feng-Ling Qing*  

        Org. Lett.2012, 14, 2870-2873. DOI: 10.1021/ol301113 

12-5: Iron-catalyzed cross-coupling reactions between arylzinc reagents and alkyl halides bearing β-fluorines 

       Xiaowei Lin, Feng Zheng, andFeng-Ling Qing*

        Organometallics2012, 31,1578-1582. DOI: 10.1021/om2005904

12-4: Copper-catalyzed aerobic oxidative trifluoromethylation of H-phosphonates using trimethyl(trifluoromethyl)silane

       Lingling Chu andFeng-Ling Qing*

        Synthesis2012, 44,1521-1525. DOI: 10.1055/2-0031-1290806

12-3: Asymmetric synthesis of β-aryl-β-trifluoromethyl-β-aminoarones via Mannich-type reactions of ketone enolates with chiral aryl CF3-substituted N-tert-butanesulfinyl ketimines

       Yingle Liu, Yangen Huang, andFeng-Ling Qing*

        Tetrahedron2012, 68,4955-4961. DOI: 10.1016/j.tet.2012.04.070

  

12-2: Synthesis and biological evaluation of SGLT2 inhibitors: gem-difluoromethylenated Dapagliflozin analogs

       Zeng-Hao Chen, Ruo-Wen Wang, andFeng-Ling Qing*

        Tetrahedron Lett.2012, 53,2171-2176. DOI: 10.1016/j.tetlet.2012.02.062 

12-1: Synthesis of γ-fluoroalkylated allylic amine derivatives via palladium-catalyzed Overman rearrangement 

       Xin-Yi Jiang, lingling Chu, Ruo-Wen Wang and Feng-Ling Qing*  

        Tetrahedron Lett.2012, 53,6853-6857. DOI: 10.1016/j.tetlet.2012.10.045

上一篇:2013年论文
返回

版权所有:中国科学院上海有机化学研究所        沪ICP备05005485号-1

地址: 上海市零陵路345号    邮政编码:200032

>